Results for:
"
Agonist
" in Documents
- Radiolabelling of the human 5-HT2A receptor with an agonist, a partial...
- Previous work has shown that 5-hydroxytryptamine (5-HT)2A receptors can be radiolabelled with various radioligands, including partial agonists, such as [125I]-DOI and [3H]-DOB, and antagonists, such a...
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Uploaded: 1996-1-12
- Short-term inverse-agonist treatment induces reciprocal changes in del...
- This study assessed the effects of short-term treatment (30-min) with inverse agonists on receptor protein levels and on the ability of agonists, inverse agonists, and neutral antagonists to bind to t...
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Uploaded: 2001-9-20
- Agonist and inverse agonist actions of beta-blockers at the human beta...
- Beta-blockers have beneficial effects in heart failure, although the underlying mechanism is unknown. Beta2-adrenoceptors, however, are proportionally higher in the failing human heart. This study sho...
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Uploaded: 2003-12-3
- Reciprocal regulation of agonist and inverse agonist signaling efficac...
- Rapid regulation of receptor signaling by agonist ligands is widely accepted, whereas short-term adaptation to inverse agonists has been little documented. In the present study, guanosine 5'-O-(3-[(35...
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Uploaded: 2004-10-22
- Mass quantitation of agonist-induced arachidonate release and icosanoi...
- The mass of total arachidonate released from phospholipids upon agonist stimulation of the cell and the fraction of released arachidonate which is converted to icosanoids are two parameters of arachid...
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Uploaded: 1988-11-5
- In vitro characterization of agonist, antagonist, inverse agonist and ...
- The efficacy of coupling between the benzodiazepine receptor and chloride channel as well as the coupling to the GABA receptor is differentially affected by different benzodiazepine ligands. In genera...
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Uploaded: 1984-1-1
- Combination of a delta opioid receptor agonist but not a mu opioid rec...
- The effects of intracerebroventricular injections of opioid peptides selective for mu or delta opioid receptors on behaviors induced by the D1 dopamine agonist SKF 38393 were investigated by using mul...
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Uploaded: 1992-3-17
- Spinal analgesia: comparison of the mu agonist morphine and the kappa ...
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Uploaded: 1981-5-11